Perphenazine-d6 (fumarate)
Perphenazine-d6 (fumarate) is a deuterated labeled Perphenazine[1]. Perphenazine is an orally active dopamine receptor and histamine-1 receptor antagonist, with Ki values of 0.56 nM (D2), 0.43 nM (D3), 6 nM (5-HT2A), respectively. Perphenazine also binds to Alpha-1A adrenergic receptor. Perphenazine inhibits cancer cell proliferation, and induces apoptosis. Perphenazine can be used in the research of mental disease, cancer, inflammation[2][4][6].
Product Specifications
CAS Number
1261432-36-3
UNSPSC
12352005
Target
5-HT Receptor; Adrenergic Receptor; Apoptosis; Autophagy; Dopamine Receptor; Histamine Receptor; Isotope-Labeled Compounds
Type
Isotope-Labeled Compounds
Related Pathways
Apoptosis; Autophagy; GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling; Others
Applications
COVID-19-immunoregulation
Field of Research
Cancer
Smiles
OC(/C=C/C(O)=O)=O.OCCN(CC1)CCN1C([2H])([2H])C([2H])([2H])C([2H])([2H])N2C3=CC(Cl)=CC=C3SC4=CC=CC=C42
Molecular Formula
C25H24D6ClN3O5S
Molecular Weight
526.08
References & Citations
Shipping Conditions
Room temperature
Scientific Category
Isotope-Labeled Compounds
Clinical Information
No Development Reported
Isoform
5-HT2 Receptor
Frequently Asked Questions
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