CPSA
Product Specifications
UNSPSC Description
CPSA is a potent and competitive inhibitor against 20α-hydroxysteroid dehydrogenase (AKR1C1) with a Ki value of 0.86 nM. CPSA is promising for research of lung and endometrial cancers, premature birth and neuronal disorders[1].
Target Antigen
Aldose Reductase; Others
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease;Others
Applications
Cancer-programmed cell death
Field of Research
Cancer; Neurological Disease
Assay Protocol
https://www.medchemexpress.com/cpsa.html
Smiles
O=C(C1=CC(C2=CC=CC=C2)=CC(Cl)=C1O)O
Molecular Weight
248.66
References & Citations
[1]El-Kabbani O, et al. Probing the inhibitor selectivity pocket of human 20α-hydroxysteroid dehydrogenase (AKR1C1) with X-ray crystallography and site-directed mutagenesis. Bioorg Med Chem Lett. 2011 Apr 15;21(8):2564-7.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-113850/CPSA-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-113850/
Clinical Information
No Development Reported
CAS Number
1038713-54-0
Curated Selection
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