CYB210010
Product Specifications
UNSPSC Description
CYB210010 is an orally bioavailable, long-acting serotonin 5-HT2 receptor agonist that selectively targets 5-HT2A and 5-HT2C receptors (EC50: 4.1 n, 7.3 nM). CYB210010 can enter the central nervous system, cause a head twitch response (HTR), and is not prone to behavioral tolerance during chronic administration[1].
Target Antigen
5-HT Receptor; Androgen Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein;Neuronal Signaling;Vitamin D Related/Nuclear Receptor
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/cyb210010.html
Solubility
10 mM in DMSO
Smiles
COC1=C(CCN)C=C(OC)C(SC(F)(F)F)=C1.Cl
Molecular Weight
317.76
References & Citations
[1]Varty GB, et al. Synthesis and Structure-Activity Relationships of 2,5-Dimethoxy-4-Substituted Phenethylamines and the Discovery of CYB210010: A Potent, Orally Bioavailable and Long-Acting Serotonin 5-HT2 Receptor Agonist. J Med Chem. 2024 Apr 25;67(8):6144-6188.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-162423/CYB210010-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-162423/
Clinical Information
No Development Reported
CAS Number
2762568-47-6
Curated Selection
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