LB30057
LB30057 (CI-1028) is an orally active selective thrombin inhibitor with an IC50 value of 0.38 nM for human thrombin. LB30057 can be used in the study of the thrombus model[1].
Product Specifications
CAS Number
184770-78-3
Product Name Alternative
CI-1028; PD 172524
UNSPSC
12352005
Target
Thrombin
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/lb30057.html
Smiles
NNC(C(C=C1)=CC=C1C[C@H](NS(=O)(C2=CC3=C(C=CC=C3)C=C2)=O)C(N(C4CCCC4)C)=O)=N
Molecular Formula
C26H31N5O3S
Molecular Weight
493.62
References & Citations
[1]Oh YS, et al. Discovery of LB30057, a benzamidrazone-based selective oral thrombin inhibitor. Bioorg Med Chem Lett. 1998 Mar 17;8 (6) :631-4.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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