DprE1-IN-11
DprE1-IN-11 (compound 3) is an orally active DprE1 inhibitor with antituberculosis activity against MTB H37Rv and MDR-MTB strains (MIC [1].
Product Specifications
UNSPSC
12352005
Target
Bacterial
Type
Reference compound
Related Pathways
Anti-infection
Field of Research
Infection
Assay Protocol
https://www.medchemexpress.com/dpre1-in-11.html
Smiles
NCCO/N=C1CCC(CC\1)CN2CCN(CC2)C3=NC(C4=CC(C(F)(F)F)=CC([N+]([O-])=O)=C4S3)=O
Molecular Formula
C22H27F3N6O4S
Molecular Weight
528.55
References & Citations
[1] Zhong X, et al. Design, synthesis and antimycobacterial activity of novel benzothiazinones with improved water solubility. Eur J Med Chem. 2024 Sep 3;279:116829.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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