(D-Arg2, Sar 4) -Dermorphin (1-4)
(D-Arg2, Sar 4) -Dermorphin (1-4) is a tetrapeptide derivative of the peptide Dermorphin found in amphibian skin. (D-Arg2, Sar 4) -Dermorphin (1-4) has significant analgesic effects by binding to the μ-opioid receptor (MOR) in the body. (D-Arg2, Sar 4) -Dermorphin (1-4) can be used in the development of analgesic drugs[1].
Product Specifications
CAS Number
90549-86-3
UNSPSC
12352209
Target
Opioid Receptor
Type
Peptides
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/d-arg2-sar-4-dermorphin-1-4.html
Smiles
OC1=CC=C(C[C@@H](C(N[C@@H](C(N[C@@H](CC2=CC=CC=C2)C(N(CC(O)=O)C)=O)=O)CCCNC(N)=N)=O)N)C=C1
Molecular Formula
C27H37N7O6
Molecular Weight
555.63
References & Citations
[1]Nakata N, et al. Physical dependence of a dermorphin tetrapeptide analog, [D-Arg2, Sar4]-dermorphin (1–4) in the rat[J]. Pharmacology Biochemistry and Behavior, 1986, 24 (1) : 27-31.
Shipping Conditions
Room temperature
Scientific Category
Peptides
Clinical Information
No Development Reported
Frequently Asked Questions
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