Risotilide
Risotilide is an inhibitor of enkephalinase B, which has the ability to inhibit enkephalinase B activity (IC50 value is 0.35 microM), and can also effectively inhibit enkephalinase A (IC50 = 0.02 microM) and aminopeptidase activity (IC50 = 13 microM), and can be regarded as a complete inhibitor of enkephalin biodegradation.
Product Specifications
CAS Number
[120688-08-6]
UNSPSC
12352005
Target
Neprilysin
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/risotilide.html
Smiles
O=S(C1=CC=C(C=C1)NS(=O)(C)=O)(N(CCNC(C)C)C(C)C)=O
Molecular Formula
C15H27N3O4S2
Molecular Weight
377.52
References & Citations
[1]Electrophysiological effects of left ventricular hypertrophy. Effect of calcium and potassium channel blockade
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Phase 2
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