β2AR antagonist 1
β2AR antagonist 1 (Cmpd-15PA) is an antagonist of β2 adrenergic receptor (β2AR) . β2AR antagonist 1 binds to the intracellular surface of the β2AR[1].
Product Specifications
CAS Number
[2135743-21-2]
UNSPSC
12352005
Target
Adrenergic Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/β2ar-antagonist-1.html
Smiles
NC(C(C=C1)=CC=C1C[C@@H](C(N[C@H](C(NCCOCCOCCOCC(O)=O)=O)CC2=CC(Br)=CC=C2)=O)NC(C(C3=CC=CC=C3)C4CCCCC4)=O)=O
Molecular Formula
C41H51BrN4O9
Molecular Weight
823.77
References & Citations
[1]Liu X, et al. Mechanism of intracellular allosteric β2AR antagonist revealed by X-ray crystal structure. Nature. 2017 Aug 24;548 (7668) :480-484.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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