Acetalin-3
Acetalin-3 (Ac-RFMWMT-NH2), a hexapeptide, is a μ opioid receptor antagonist with high affinity for μ and κ3 opioid receptor, weak affinity for κ1 receptors and no affinity for κ2 receptors[1].
Product Specifications
CAS Number
152274-65-2
UNSPSC
12352209
Target
Opioid Receptor
Type
Peptides
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/acetalin-3.html
Solubility
10 mM in DMSO
Smiles
C[C@@H](O)[C@@H](C(N)=O)NC([C@H](CCSC)NC([C@@H](NC([C@H](CCSC)NC([C@@H](NC([C@@H](NC(C)=O)CCCNC(N)=N)=O)CC1=CC=CC=C1)=O)=O)CC2=CNC3=CC=CC=C23)=O)=O
Molecular Formula
C42H61N11O8S2
Molecular Weight
912.13
References & Citations
[1]C T Dooley, et al. Acetalins: opioid receptor antagonists determined through the use of synthetic peptide combinatorial libraries. Proc Natl Acad Sci U S A. 1993 Nov 15;90 (22) :10811-5.
Shipping Conditions
Room temperature
Scientific Category
Peptides
Clinical Information
No Development Reported
Isoform
μ Opioid Receptor/MOR
Frequently Asked Questions
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