BigLEN (mouse) (TFA)

BigLEN (mouse) TFA is a GPR171 agonist. BigLEN (mouse) TFA is a proSAAS-derived neuropeptide. BigLEN (mouse) TFA regulates food intake in mice. BigLEN (mouse) inhibits the release of glutamate onto parvocellular neurons of the paraventricular nucleus in a process dependent upon activation of postsynaptic G proteins.

Product Specifications

UNSPSC

12352209

Target

GPR171

Type

Peptides

Related Pathways

GPCR/G Protein

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/biglen-mouse-tfa.html

Solubility

10 mM in DMSO

Smiles

O=C(N1[C@@H](CCC1)C(O)=O)[C@H]2N(CCC2)C([C@H](CC(C)C)NC([C@H](CC(C)C)NC([C@H](CCCNC(N)=N)NC([C@H](CCCNC(N)=N)NC([C@H](C)NC([C@H]3N(CCC3)C([C@H](C)NC([C@H](CCC(N)=O)NC([C@H]4N(CCC4)C([C@H](CO)NC([C@H]5N(CCC5)C([C@H](CC(N)=O)NC([C@H](CCC(O)=O)NC([C@@H](N)CC(C)C)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O.O=C(C(F)(F)F)O