MerTK-IN-1
MerTK-IN-1 (compund 31) is a MerTK inhibitor with in vivo target binding ability[1].
Product Specifications
CAS Number
3036376-10-7
UNSPSC
12352005
Target
TAM Receptor
Type
Reference compound
Related Pathways
Protein Tyrosine Kinase/RTK
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/mertk-in-1.html
Smiles
NC(C1=C(N=CC(C2CN(C2)C3=NC4=C(O3)C=C(OCC(C)(O)C)C=C4)=N1)NC5=CN(N=C5)C)=O
Molecular Formula
C23H26N8O4
Molecular Weight
478.50
References & Citations
[1]Frey RR, et al. Discovery of Potent Azetidine-Benzoxazole MerTK Inhibitors with In Vivo Target Engagement. J Med Chem. 2024 Oct 10;67 (19) :17033-17052.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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