GPR109 receptor agonist-2
GPR109 receptor agonist-2 (Compound 5) is a selective GPR109a agonist with a pEC50 of 5.53[1].
Product Specifications
CAS Number
[957129-38-3]
UNSPSC
12352005
Hazard Statement
H315, H319, H335
Target
GPR109A
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/gpr109-receptor-agonist-2.html
Concentration
10mM
Purity
99.08
Solubility
DMSO : 200 mg/mL (ultrasonic)
Smiles
O=C(O)C1=NNC(CC)=C1C
Molecular Formula
C7H10N2O2
Molecular Weight
154.17
Precautions
H315, H319, H335
References & Citations
[1]Skinner PJ, et al. Fluorinated pyrazole acids are agonists of the high affinity niacin receptor GPR109a. Bioorg Med Chem Lett. 2007 Oct 15;17 (20) :5620-3.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Curated Selection
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