Dazcapistat
Dazcapistat is a potent calpain inhibitor, with IC50s of [1].
Product Specifications
CAS Number
2221010-42-8
Product Name Alternative
BLD-2660
UNSPSC
12352005
Target
Proteasome
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/dazcapistat.html
Purity
98.0
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
O=C(C(C(CC1=CC=CC=C1)NC(C2=C(C3=C(F)C=CC=C3)N=C(C)O2)=O)=O)N
Molecular Formula
C21H18FN3O4
Molecular Weight
395.38
References & Citations
[1]Brad Owen BUCKMAN, et al. Calpain modulators and therapeutic uses thereof. WO2018064119A1.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
Phase 2
Available Sizes
Frequently Asked Questions
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