MI-1544

MI-1544 is a powerful GnRH antagonist. MI-1544 induces inhibitory effects on the pituitary LH release and on gonads. MI-1544 can be used for the research of antifertility effect[1].

Product Specifications

CAS Number

[87565-51-3]

UNSPSC

12352209

Target

GnRH Receptor

Type

Peptides

Related Pathways

GPCR/G Protein

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Metabolic Disease

Assay Protocol

https://www.medchemexpress.com/mi-1544.html

Solubility

10 mM in DMSO

Smiles

ClC(C=C1)=CC=C1C[C@@H](NC([C@H](NC(C)=O)CC2=CNC3=CC=CC=C23)=O)C(N[C@@H](C(N[C@@H](CO)C(N[C@H](C(N[C@H](CCCCN)C(N[C@@H](CC(C)C)C(N[C@@H](CCCNC(N)=N)C(N4[C@@H](CCC4)C(N[C@H](C)C(N)=O)=O)=O)=O)=O)=O)CC5=CC=C(C=C5)O)=O)=O)CC6=CNC7=CC=CC=C67)=O

Molecular Formula

C71H94ClN17O13

Molecular Weight

1429.07

References & Citations

[1]Kovács M, et al. Effects of long-term administration of a superactive agonistic and an antagonistic GnRH analog on the pituitary-gonad system. Peptides. 1989 Sep-Oct;10 (5) :925-31.