APD-916
APD-916 is an H3 receptor antagonist. APD-916 shows good pharmacokinetic properties, and oral administration of APD-916 has been shown to enhance wakefulness in various animal models[1].
Product Specifications
CAS Number
[1021169-11-8]
UNSPSC
12352005
Target
Histamine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/apd-916.html
Smiles
C[C@H]1N(CCC2=CC=C(C3=CC=C(S(=O)(CCCOC)=O)C=C3)C=C2)CCC1
Molecular Formula
C23H31NO3S
Molecular Weight
401.56
References & Citations
[1]Ghamari N, et al. Histamine H3 receptor antagonists/inverse agonists: Where do they go? Pharmacol Ther. 2019 Aug;200:69-84.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Phase 1
Curated Selection
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