PGN-9856
Product Specifications
Product Name Alternative
2-Octadecyl-1H-indole-5-carboxylic acid
UNSPSC Description
PGN-9856 is a selective and high affinity (pKi ≥ 8.3) ligand at EP2 receptor. PGN-9856 is a potetn and non-prostanoid EP2 receptor agonist (pEC50 ≥ 8.5). PGN-9856 shows anti-inflammatory and anti-glaucoma activities[1].
Target Antigen
Prostaglandin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/pgn-9856.html
Purity
98.90
Solubility
DMSO : 125 mg/mL (ultrasonic)
Smiles
O=C(O)COC1=CC=CC(NC(C2=CC(C3=CC=CC(F)=C3)=CC=C2F)=O)=C1
Molecular Weight
383.34
References & Citations
[1]Coleman RA, et al. The affinity, intrinsic activity and selectivity of a structurally novel EP2 receptor agonist at human prostanoid receptors. Br J Pharmacol. 2019 Mar;176(5):687-698.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C, 3 years (Powder)
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-115462/PGN-9856-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-115462/PGN-9856-SDS-MedChemExpress.pdf
Clinical Information
No Development Reported
CAS Number
863704-91-0
Available Sizes
Curated Selection
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