(Rac) -Enadoline
(Rac) -Enadoline ((Rac) -CI-977 free base) is a selective K-opioid receptor agonist that stereoselectively antagonizes clonic seizures induced by slow intravenous injection of N-methyl-DL-aspartate in mice[1].
Product Specifications
CAS Number
[107431-28-7]
Product Name Alternative
(Rac) -CI-977 (free base)
UNSPSC
12352005
Target
Opioid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/rac-enadoline.html
Smiles
O=C(CC1=CC=CC2=C1C=CO2)N(C3C(N4CCCC4)CC5(CCCO5)CC3)C
Molecular Formula
C24H32N2O3
Molecular Weight
396.52
References & Citations
[1]Singh L, et al. The anticonvulsant action of CI-977, a selective κ-opioid receptor agonist: a possible involvement of the glycine/NMDA receptor complex[J]. European journal of pharmacology, 1990, 191 (3) : 477-480.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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