[Nphe1]Nociceptin (1-13) NH2 (TFA)
[Nphe1]Nociceptin (1-13) NH2, a novel nociceptin/orphanin FQ (NC) endogenous ligand, is a selective and competitive ociceptin receptor antagonist without any residual agonist activity. [Nphe1]nociceptin (1-13) NH2 binds selectively to recombinant nociceptin receptors (pKi=8.4) and antagonizes the inhibitory effects of nociceptin on cyclic AMP accumulation in CHO cells (pA2=6.0) . [Nphe1]Nociceptin (1-13) NH2 has the potential to act as an analgesic agent[1].
Product Specifications
UNSPSC
12352209
Target
Opioid Receptor
Type
Peptides
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/nphe1-nociceptin-1-13-nh2-tfa.html
Solubility
10 mM in DMSO
Smiles
Molecular Formula
C63H101F3N22O17
Molecular Weight
1495.61
References & Citations
Shipping Conditions
Room temperature
Scientific Category
Peptides
Clinical Information
No Development Reported
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