Mazisotine
SSTR4 agonist-1 (Compound 47) is a selective agonist for somatostatin receptor subtype 4 (SSTR4) with an EC50 of 4.7 nM. SSTR4 agonist-1 reveals a half-life > 130 minutes in human liver microsomes[1].
Product Specifications
CAS Number
[1638588-92-7]
UNSPSC
12352005
Hazard Statement
H302, H315, H319, H335
Target
Somatostatin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology; Neurological Disease
Assay Protocol
https://www.medchemexpress.com/sstr4-agonist-1.html
Purity
99.54
Solubility
DMSO : 125 mg/mL (ultrasonic)
Smiles
CC(C=CC=N1)=C1OCC(C)(C)NC([C@H]2[C@@]3([H])[C@]2([H])CNC3)=O
Molecular Formula
C16H23N3O2
Molecular Weight
289.37
Precautions
H302, H315, H319, H335
References & Citations
[1]Giovannini R, et al., New somatostatin receptor subtype 4 (sstr4) agonists. WO2014184275 A1.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
SSTR4
Available Sizes
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