(-) -Dihydroalprenolol

(-) -Dihydroalprenolol (L-Dihydroalprenolol) is a β-adrenergic antagonist that inhibits the activity of β-adrenergic receptors. (-) -Dihydroalprenolol can cause desensitization of approximately 60% of β-adrenergic receptor binding sites. (-) -Dihydroalprenolol has also been shown to reduce the binding capacity of specific β-adrenergic ligands. (-) -Dihydroalprenolol may affect the ability to stimulate membrane-bound adenylate acylase[1].

Product Specifications

CAS Number

[59624-90-7]

Product Name Alternative

L-Dihydroalprenolol

UNSPSC

12352005

Target

Adrenergic Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Endocrinology

Assay Protocol

https://www.medchemexpress.com/minus-dihydroalprenolol.html

Concentration

10mM

Purity

99.63

Solubility

DMSO : 100 mg/mL (ultrasonic)

Smiles

O[C@@H](CNC(C)C)COC1=CC=CC=C1CCC

Molecular Formula

C15H25NO2

Molecular Weight

251.36

References & Citations

[1]Desensitization of beta-adrenergic receptors by beta-adrenergic agonists in a cell-free system: resensitization by guanosine 5'- (beta, gamma-imino) triphosphate and other purine nucleotides