Eptapirone (fumarate)
Eptapirone fumarate (F11440 fumarate) is a potent, selective and orally active 5-HT1A receptor agonist (pKi = 8.33) . Eptapirone fumarate can inhibit cAMP production. Eptapirone fumarate can reduce 5-HT levels and increase corticosterone levels. Eptapirone fumarate shows potent anxiolytic and antidepressant potential. Eptapirone fumarate can be used for the research of neurological disease, such as anxiety and depression[1].
Product Specifications
CAS Number
179756-85-5
Product Name Alternative
F 11440 (fumarate)
UNSPSC
12352005
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/eptapirone-fumarate.html
Smiles
O=C(O)/C=C/C(O)=O.O=C(N1C)N(CCCCN2CCN(C3=NC=CC=N3)CC2)N=CC1=O
Molecular Formula
C20H27N7O6
Molecular Weight
461.47
References & Citations
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Phase 1
Isoform
5-HT1 Receptor
Frequently Asked Questions
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