Rociverine
Product Specifications
UNSPSC Description
Rociverine is an anticholinergic compound with smooth muscle relaxant activity. Rociverine showed different binding modes in five cloned muscarinic receptors. The cis stereoisomer of Rociverine showed a higher affinity change compared to the trans stereoisomer. The (1R,2R) configuration of Rociverine showed significantly higher affinity, even up to 240 times. The (1S,2S) configuration of Rociverine is very important for binding selectivity[1].
Target Antigen
Endogenous Metabolite
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/rociverine.html
Smiles
O[C@@]1(C2CCCCC2)[C@H](CCCC1)C(OC(C)CN(CC)CC)=O
Molecular Weight
339.51
References & Citations
[1]Stereoselective inhibition of muscarinic receptor subtypes by the eight stereoisomers related to rociverine
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-122294/Rociverine-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-122294/
Clinical Information
No Development Reported
CAS Number
53716-44-2
Curated Selection
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