LDN-209929
LDN-209929 is a potent haspin kinase inhibitor, with IC50 values of 55 nM and 9.9 μM for Haspin and DYRK2, respectively[1].
Product Specifications
CAS Number
1233355-57-1
UNSPSC
12352005
Target
Haspin Kinase
Type
Reference compound
Related Pathways
Cell Cycle/DNA Damage
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/ldn-209929.html
Smiles
ClC1=CC2=C(N=C3C=CC(OC)=CC3=C2SCCCN)C=C1
Molecular Formula
C17H17ClN2OS
Molecular Weight
332.85
References & Citations
[1]Gregory D Cuny, et al. Structure-activity relationship study of acridine analogs as haspin and DYRK2 kinase inhibitors. Bioorg Med Chem Lett. 2010 Jun 15;20 (12) :3491-4.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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