17β-HSD5 inhibitor 3
17β-HSD5 inhibitor 3 (Compound 31) is an orally active inhibitor for 17β-HSD5 with an IC50 of 69 nM[1].
Product Specifications
CAS Number
948581-46-2
UNSPSC
12352005
Target
17β-HSD
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/17β-hsd5-inhibitor-3.html
Smiles
O=C(O)C1=CN(S(=O)(C2=CC=C(Br)C=C2)=O)C3=C(Cl)C=CC=C31
Molecular Formula
C15H9BrClNO4S
Molecular Weight
414.66
References & Citations
[1]Marchais-Oberwinkler S, et al., 17β-Hydroxysteroid dehydrogenases (17β-HSDs) as therapeutic targets: protein structures, functions, and recent progress in inhibitor development. J Steroid Biochem Mol Biol. 2011 May;125 (1-2) :66-82.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
KHK-C
Frequently Asked Questions
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