Apimostinel
Apimostinel (NRX-1074; AGN-241660) is an orally active NMDA receptor partial agonist[1].
Product Specifications
CAS Number
[1421866-48-9]
Product Name Alternative
NRX-1074; AGN-241660
UNSPSC
12352005
Target
IGluR
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neurodegeneration
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/Apimostinel.html
Purity
99.04
Solubility
DMSO : 155 mg/mL (ultrasonic) |H2O : ≥ 6.67 mg/mL
Smiles
C[C@@H](O)[C@@H](C(N)=O)NC([C@@]1(CC2=CC=CC=C2)N(C([C@H]3N(C([C@H]([C@H](O)C)N)=O)CCC3)=O)CCC1)=O
Molecular Formula
C25H37N5O6
Molecular Weight
503.59
References & Citations
[1]Naurex's First Orally Active Molecule, NRX-1074, Demonstrates Statistically Significant Improvement in Depression Scores within 24 Hours in Phase 2 Study for Major Depressive Disorder. January 28, 2015.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, stored under nitrogen)
Scientific Category
Reference compound1
Clinical Information
Phase 2
Isoform
NMDA Receptor
Available Sizes
Curated Selection
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