PCSK9-IN-26
PCSK9-IN-26 (Compound 116) is an PCSK9 inhibitor (IC50 [1].
Product Specifications
CAS Number
[3033361-09-7]
UNSPSC
12352005
Target
PCSK9
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/pcsk9-in-26.html
Solubility
10 mM in DMSO
Smiles
O=C1N(C(C=C(C#N)C=C2)=C2N1C)C3=CC=C(N[C@@H]4C[C@@H](NC5=NC=C(C6CC6)N=N5)CC4)N=C3
Molecular Formula
C25H25N9O
Molecular Weight
467.53
References & Citations
[1]Gavin D, et al. Pcsk9 inhibitors and methods of use thereof, WO2024062090A1, 2024
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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