AS2717638
AS2717638 is a highly selective, brain-penetrant and orally active lysophosphatidic acid receptor 5 (LPA5) antagonist with an IC50 value of 38 nM. AS2717638 is highly selective and shows no significant antagonistic activity against other LPA receptors (LPA1, LPA2, and LPA3) . AS2717638 can be used in the research of pain and neuroinflammation-related diseases[1][2].
Product Specifications
CAS Number
2148339-28-8
Product Name Alternative
OPC-14857 (Standard); DM-14857 (Standard),OPC-14857; DM-14857
UNSPSC
12352005
Target
LPL Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Inflammation/Immunology; Neurological Disease
Assay Protocol
https://www.medchemexpress.com/AS2717638.html
Purity
99.85
Solubility
DMSO : 60 mg/mL (ultrasonic)
Smiles
O=C1N(C=C(C2=C1C=C(C(OC)=C2)OC)C(N3CCCCC3)=O)C4=NOC5=C4C=C(C=C5)C
Molecular Formula
C25H25N3O5
Molecular Weight
447.48
References & Citations
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
LPAR5
Available Sizes
Frequently Asked Questions
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