GPR84 antagonist 1
GPR84 antagonist 1 is a high affinity and highly selective competitive antagonist of human GPR84.
Product Specifications
CAS Number
[2762180-28-7]
UNSPSC
12352005
Target
GPR84
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/gpr84-antagonist-1.html
Purity
98.56
Solubility
DMSO : 50 mg/mL (ultrasonic)
Smiles
COC1=CC=C(C2=C(C3=CC=C(OC)C=C3)N=C(CC4=CNC5=C4C=CC=C5)N=N2)C=C1
Molecular Formula
C26H22N4O2
Molecular Weight
422.48
References & Citations
[1]Jenkins L, et al. Discovery and Characterization of Novel Antagonists of the Proinflammatory Orphan Receptor GPR84. ACS Pharmacol Transl Sci. 2021 Sep 7;4 (5) :1598-1613.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Curated Selection
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