TBPC

TBPC is a selective positive allosteric modulator for human Y4 receptor (Y4R), which enhances the activation of Y4R in G protein signaling and arrestin3 recruitment[1].

Product Specifications

CAS Number

[1942-71-8]

UNSPSC

12352005

Hazard Statement

H302, H315, H319, H335

Target

Neuropeptide Y Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Metabolic Disease

Assay Protocol

https://www.medchemexpress.com/tbpc.html

Purity

98.41

Solubility

DMSO : 100 mg/mL (ultrasonic)

Smiles

OC1C(OC2=CC=C(C(C)(C)C)C=C2)CCCC1

Molecular Formula

C16H24O2

Molecular Weight

248.36

Precautions

H302, H315, H319, H335

References & Citations

[1]Schubert M, et al., Identification and Characterization of the First Selective Y4 Receptor Positive Allosteric Modulator. J Med Chem. 2017 Sep 14;60 (17) :7605-7612.