H4R antagonist 3

H4R antagonist 3 (Example 18) is a histamine-4 receptor antagonist with an EC50 of [1].

Product Specifications

CAS Number

[1003091-20-0]

UNSPSC

12352005

Target

Histamine Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling

Applications

COVID-19-immunoregulation

Field of Research

Inflammation/Immunology

Assay Protocol

https://www.medchemexpress.com/h4r-antagonist-3.html

Purity

96.29

Solubility

DMSO : 2 mg/mL (ultrasonic; warming; heat to 60°C)

Smiles

ClC1=CC=C(C2=CSC3=NC=NC(N(C4CCN(CC4)C)C)=C32)C=C1

Molecular Formula

C19H21ClN4S

Molecular Weight

372.91

References & Citations

[1]Allen J. Borchardt, et al. Aminopyrimidine inhibitors of histamine receptors for the treatment of disease. Patent US20100063047A1.

Shipping Conditions

Room Temperature

Storage Conditions

4°C (Powder, protect from light)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Available Sizes

Curated Selection

Explore Other Products

Discover premium biology products from our extensive collection of 20M+ items

MBS1275854-01 0.01 mg Plasmid + 0.2 mL Glycerol-Stock

CACNG1 cDNA Clone

Ask

View Details

MBS1275854-02 5x 0.01 mg Plasmid + 5x 0.2 mL Glycerol-Stock

CACNG1 cDNA Clone

Ask

View Details

MBS6470541-01 0.1 mL

CKMM, NT (Creatine Kinase M-type, Creatine Kinase M Chain, M-CK, CKM) (MaxLight 550)

Ask

View Details

MBS6470541-02 5x 0.1 mL

CKMM, NT (Creatine Kinase M-type, Creatine Kinase M Chain, M-CK, CKM) (MaxLight 550)

Ask

View Details

ABC-KD1408 1 Vial

Human BCS1L knockdown cell line

Ask

View Details

VCar-Ly227 5 mg

Vitamin D PEG (2 kDa)

Ask

View Details