SKF 100398

SKF 100398 (d (CH2) 5Tyr (Et) VAVP), an arginine vasopressin (AVP) analogue, is a specific antagonist of the antidiuretic effect of exogenous and endogenous AVP[1].

Product Specifications

CAS Number

[77453-01-1]

Product Name Alternative

D (CH2) 5Tyr (Et) VAVP

UNSPSC

12352209

Hazard Statement

H332

Target

Vasopressin Receptor

Type

Peptides

Related Pathways

GPCR/G Protein

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Metabolic Disease

Assay Protocol

https://www.medchemexpress.com/skf-100398.html

Purity

99.48

Solubility

10 mM in DMSO

Smiles

O=C(N[C@@H](CCCNC(N)=N)C(NCC(N)=O)=O)[C@H]1N(C([C@@H](NC([C@H](CC(N)=O)NC([C@H](C(C)C)NC([C@H](CC2=CC=CC=C2)NC3=O)=O)=O)=O)CSSC4(CCCCC4)CC(N[C@H]3CC5=CC=C(OCC)C=C5)=O)=O)CCC1

Molecular Formula

C53H77N13O11S2

Molecular Weight

1136.39

Precautions

H332

References & Citations

[1]S Ishikawa, et al. Further in vivo evidence for antagonist-to-antidiuretic action of arginine vasopressin. Am J Physiol. 1983 Nov;245 (5 Pt 1) :R713-9.