CYT-1010 (hydrochloride)
CYT-1010 hydrochloride is a mu-opioid receptor agonist extracted from patent WO2013173730A2, with EC50s of 13.1 nM and 0.0053 nM on beta-arrestin recruitment and inhibition of cAMP production, respectively[1].
Product Specifications
CAS Number
1161517-81-2
UNSPSC
12352005
Target
Opioid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/cyt-1010-hydrochloride.html
Solubility
10 mM in DMSO
Smiles
OC1=CC=C(C=C1)C[C@@H](C(N[C@H](CCCCNC2=O)C(N[C@@H](CC3=CNC4=C3C=CC=C4)C(N[C@H]2CC5=CC=CC=C5)=O)=O)=O)N.Cl
Molecular Formula
C35H41ClN6O5
Molecular Weight
661.19
References & Citations
[1]Theodore E. Maione, Novel therapeutic uses of mu-opiate receptor peptides. WO2013173730A2.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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