Gabazine (free base)
Gabazine is a selective and competitive antagonist of GABAA receptor, with an IC50 of 0.2 μM for GABA receptor[1].
Product Specifications
CAS Number
[105538-73-6]
Product Name Alternative
SR95531 (free base)
UNSPSC
12352005
Target
GABA Receptor
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/gabazine-free-base.html
Smiles
O=C(CCCN1N=C(C2=CC=C(OC)C=C2)C=CC1=N)O
Molecular Formula
C15H17N3O3
Molecular Weight
287.31
References & Citations
[1]Ueno S, et al. Bicuculline and gabazine are allosteric inhibitors of channel opening of the GABAA receptor. J Neurosci. 1997 Jan 15;17 (2) :625-34.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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