PKCη pseudosubstrate inhibitor, myristoylated

PKCη pseudosubstrate inhibitor, myristoylated is cell permeable and can be used to study the mechanism of action of PKCη[1].

Product Specifications

CAS Number

[908012-19-1]

UNSPSC

12352209

Target

PKC

Type

Peptides

Related Pathways

Epigenetics; TGF-beta/Smad

Applications

Cancer-Kinase/protease

Field of Research

Others

Assay Protocol

https://www.medchemexpress.com/pkcη-pseudosubstrate-inhibitor-myristoylated.html

Purity

96.72

Solubility

DMSO : 100 mg/mL (ultrasonic)

Smiles

OC(CNC([C@H](CC(N)=O)NC([C@H]([C@@H](C)CC)NC([C@H](CCC(N)=O)NC([C@@H](NC([C@H](C(C)C)NC([C@H](CCCNC(N)=N)NC([C@H](CCCNC(N)=N)NC([C@H](CCCNC(N)=N)NC([C@H](CCSC)NC([C@H](C)NC([C@H](CCCNC(N)=N)NC([C@H](CCC(N)=O)NC([C@H](CCCNC(N)=N)NC([C@H](CCCCN)NC([C@H](CCCNC(N)=N)NC([C@H]([C@H](O)C)NC(CCCCCCCCCCCCC)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)CC1=CN=CN1)=O)=O)=O)=O)=O

Molecular Formula

C101H185N41O23S

Molecular Weight

2373.88

References & Citations

[1]Muzorewa TT, et al. Coordinated regulation of endothelial calcium signaling and shear stress-induced nitric oxide production by PKCβ and PKCη. Cell Signal. 2021 Nov;87:110125.