Relenopride
Relenopride is a agonist of novel potent 5-HT4 receptor partial with weak binding to 5-HT 2B receptors (Ki = 31 nM) [1].
Product Specifications
CAS Number
1221416-43-8
Product Name Alternative
YKP10811
UNSPSC
12352005
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/relenopride.html
Smiles
NC(O[C@H](C1=CC=C(C=C1)F)CCN(CC2)CCC2CNC(C3=C(C=C(C(Cl)=C3)N)OC)=O)=O
Molecular Formula
C24H30ClFN4O4
Molecular Weight
492.97
References & Citations
[1]Anna Zielińska, et al. Chronic abdominal pain in irritable bowel syndrome - current and future therapies. Expert Rev Clin Pharmacol. 2018 Jul;11 (7) :729-739.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Phase 3
Isoform
5-HT2 Receptor
Frequently Asked Questions
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