Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

Gestrinone (Standard)

Gestrinone (Standard) is the analytical standard of Gestrinone. This product is intended for research and analytical applications. Gestrinone (R2323) is a synthetic steroid hormone used to treat endometriosis. It inhibits leiomyoma cells with an IC50 of 43.67 μM. Gestrinone is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

Product Specifications

CAS Number

16320-04-0

Product Name Alternative

R 2323 (Standard)

UNSPSC

12352211

Target

Estrogen Receptor/ERR; Reference Standards

Type

Reference Standards

Related Pathways

Others; Vitamin D Related/Nuclear Receptor

Field of Research

Inflammation/Immunology

Assay Protocol

https://www.medchemexpress.com/gestrinone-standard.html

Smiles

C#C[C@]1(O)CC[C@@]2([H])[C@]3([H])CCC4=CC(CCC4=C3C=C[C@]12CC)=O

Molecular Formula

C21H24O2

Molecular Weight

308.41

References & Citations

[1]Tamaya T, et al. Gestrinone (R2323) binding to steroid receptors in human uterine endometrial cytosol. Acta Obstet Gynecol Scand. 1986;65 (5) :439-41.|[2]Zhu Y, et al. Gestrinone inhibits growth of human uterine leiomyoma may relate to activity regulation of ERα, Src and P38 MAPK. Biomed Pharmacother. 2012 Dec;66 (8) :569-77.|[3]Snyder BW, et al. Studies on the mechanism of action of danazol and gestrinone (R2323) in the rat: evidence for a masked estrogen component. Fertil Steril. 1989 Apr;51 (4) :705-10.|[4]Dowsett M, et al. A comparison of the effects of danazol and gestrinone on testosterone binding to sex hormone binding globulin in vitro and in vivo. Clin Endocrinol (Oxf) . 1986 May;24 (5) :555-63.

Shipping Conditions

Room temperature

Scientific Category

Reference Standards

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

HOXD3 Conjugated Antibody
orb1616677 100 µL

HOXD3 Conjugated Antibody

Sign In for Pricing
View Details
EPG5 Polyclonal Antibody
RA24601-01 50 µL

EPG5 Polyclonal Antibody

Sign In for Pricing
View Details
EPG5 Polyclonal Antibody
RA24601-02 100 µL

EPG5 Polyclonal Antibody

Sign In for Pricing
View Details
LymnaDFamide-1
H-1648.0005 5.0mg

LymnaDFamide-1

Sign In for Pricing
View Details
PCMV-SETD7 (human) (1-128aa) -3xFLAG-SV40-Neo
BZ45014 1 Vial

PCMV-SETD7 (human) (1-128aa) -3xFLAG-SV40-Neo

Sign In for Pricing
View Details
Anti-EIF2S3 Antibody Picoband® HRP Conjugated
A09574-1-HRP 100 µg/Vial

Anti-EIF2S3 Antibody Picoband® HRP Conjugated

Sign In for Pricing
View Details