Flibanserin-d4
Flibanserin-d4 is a deuterium labeled Flibanserin (BIMT-17) . Flibanserin is a full agonist of the serotonin 5-HT1A receptor (Ki=1 nM) and an antagonist of 5-HT2A (49 nM) [1].
Product Specifications
CAS Number
2122830-90-2
Product Name Alternative
BIMT-17-d4; BIMT-17BS-d4
UNSPSC
12352005
Target
5-HT Receptor
Type
Isotope-Labeled Compounds
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Solubility
10 mM in DMSO
Smiles
O=C1NC2=C([2H])C([2H])=C([2H])C([2H])=C2N1CCN3CCN(C4=CC=CC(C(F)(F)F)=C4)CC3
Molecular Formula
C20H17D4F3N4O
Molecular Weight
394.43
References & Citations
[1]Invernizzi RW, et al. Flibanserin, a potential antidepressant drug, lowers 5-HT and raises dopamine and noradrenaline in the rat prefrontal cortex dialysate: role of 5-HT (1A) receptors. Br J Pharmacol. 2003 Aug;139 (7) :1281-8.
Shipping Conditions
Room temperature
Scientific Category
Isotope-Labeled Compounds
Clinical Information
No Development Reported
Isoform
5-HT1 Receptor;5-HT2 Receptor
Available Sizes
Frequently Asked Questions
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