TASP0390325
Product Specifications
UNSPSC Description
TASP0390325 is a high affinity and orally active arginine vasopressin receptor 1B (V1B receptor) antagonist with antidepressant and anxiolytic activities[1].
Target Antigen
Vasopressin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Field of Research
Neurological Disease; Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/tasp0390325.html
Purity
99.0
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
O=C(CN1C(C2=CC(OCCCN3CCOCC3)=CN=C2N=C1C4=CC=C(C(Cl)=C4)F)=O)NC(C)C.Cl
Molecular Weight
554.44
References & Citations
[1]M Iijima, et al. Antidepressant and anxiolytic profiles of newly synthesized arginine vasopressin V1B receptor antagonists: TASP0233278 and TASP0390325. Br J Pharmacol. 2014 Jul;171(14):3511-25.|[2]Kazumi Koga, et al. High-Contrast PET Imaging of Vasopressin V 1B Receptors with a Novel Radioligand, <sup>11</sup>C-TASP699. J Nucl Med. 2017 Oct;58(10):1652-1658.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C (Powder, sealed storage, away from moisture)
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-117820/TASP0390325-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-117820/TASP0390325-SDS-MedChemExpress.pdf
Clinical Information
No Development Reported
CAS Number
1642187-96-9
Available Sizes
Curated Selection
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