Rupatadine (Fumarate)
Rupatadine (UR-12592) Fumarate is a potent, orally active and long-lasting dual PAF/H1 antagonist, with Kis of 0.55 μM and 0.1 μM, respectively. Rupatadine Fumarate can be used for the research of allergic rhinitis and urticaria[1][2][3].
Product Specifications
CAS Number
182349-12-8
Product Name Alternative
UR-12592 (Fumarate)
UNSPSC
12352005
Hazard Statement
H302, H413
Target
Autophagy; Histamine Receptor
Type
Reference compound
Related Pathways
Autophagy; GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/Rupatadine-Fumarate.html
Purity
99.99
Solubility
DMSO : 30 mg/mL (ultrasonic; warming)
Smiles
CC1=CN=CC(CN2CC/C(CC2)=C3C4=CC=C(Cl)C=C4CCC5=CC=CN=C5\3)=C1.O=C(O)/C=C/C(O)=O
Molecular Formula
C30H30ClN3O4
Molecular Weight
532.03
Precautions
H302, H413
References & Citations
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, sealed storage, away from moisture)
Scientific Category
Reference compound1
Clinical Information
Launched
Isoform
H1 Receptor
Citation 01
Pharmaceutics. 2020 Jun 8;12 (6) :525.|Biomed Pharmacother. 2024 Jun 4:176:116826.
Available Sizes
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