Yp537

Yp537 is an estrogen receptor (ER) inhibitor that blocks dimerization of the human estrogen receptor[1].

Product Specifications

CAS Number

[166664-90-0]

Product Name Alternative

Anti-estrogen

UNSPSC

12352209

Target

Estrogen Receptor/ERR

Type

Peptides

Related Pathways

Vitamin D Related/Nuclear Receptor

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Endocrinology

Assay Protocol

https://www.medchemexpress.com/yp537.html

Solubility

H2O

Smiles

SC[C@H](N)C(N[C@@H](CC(N)=O)C(N[C@@H](C(C)C)C(N[C@@H](C(C)C)C(N1[C@@H](CCC1)C(N[C@@H](CC(C)C)C(N[C@H](C(N[C@@H](CC(O)=O)C(N[C@@H](CC(C)C)C(N[C@@H](CC(C)C)C(N[C@@H](CC(C)C)C(N[C@H](C(O)=O)CCC(O)=O)=O)=O)=O)=O)=O)CC2=CC=C(C=C2)OP(O)(O)=O)=O)=O)=O)=O)=O)=O

Molecular Formula

C64H104N13O22PS

Molecular Weight

1470.62

References & Citations

[1]Arnold SF, et al. An antiestrogen: a phosphotyrosyl peptide that blocks dimerization of the human estrogen receptor. Proc Natl Acad Sci U S A. 1995 Aug 1;92 (16) :7475-9.