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CaMdr1p-IN-1

Product Specifications

UNSPSC Description

CaMdr1p-IN-1 (Compound A) is an inhibitor for the major facilitator superfamily transporter CaMdr1p. CaMdr1p-IN-1 exhibits chemosensitizing efficacy. CaMdr1p-IN-1 synergizes with Fluconazole (HY-B0101), that inhibits CaMdr1p overexpressing Candida albicans with MIC of 10 μM[1].

Target Antigen

Others

Type

Reference compound

Related Pathways

Others

Applications

COVID-19-immunoregulation

Field of Research

Infection

Assay Protocol

https://www.medchemexpress.com/camdr1p-in-1.html

Smiles

O=C1C(C(NC2=CC=CC=C2)=C1/C=C3N(C4=C(C\3(C)C)C=CC=C4)C)=O

Molecular Weight

344.41

References & Citations

[1]Keniya MV, et al., Inhibitors of the Candida albicans Major Facilitator Superfamily Transporter Mdr1p Responsible for Fluconazole Resistance. PLoS One. 2015 May 7;10(5):e0126350.

Shipping Conditions

Room temperature

Product Datasheet

http://file.medchemexpress.com/batch_PDF/HY-120432/CaMdr1p-IN-1-DataSheet-MedChemExpress.pdf

Product MSDS

http://file.medchemexpress.com/batch_PDF/HY-120432/

Clinical Information

No Development Reported

CAS Number

1257542-38-3

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