Legumain inhibitor 1
Legumain inhibitor 1 is a potent and selective Legumain inhibitor with an IC50 of 3.6 nM. Legumain inhibitor 1 can be used for cancer research[1].
Product Specifications
CAS Number
2361157-34-6
UNSPSC
12352005
Target
Legumain
Type
Reference compound
Related Pathways
Neuronal Signaling
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/legumain-inhibitor-1.html
Purity
99.18
Solubility
DMSO : 40 mg/mL (ultrasonic)
Smiles
O=C(N[C@H](C#N)CC(N)=O)C(C)(C)CS(=O)(C1=CC=C(C2=CC3=C(N(C)N=C3)C=C2)C=C1)=O
Molecular Formula
C23H25N5O4S
Molecular Weight
467.54
References & Citations
[1]Sharon L Eddie, et al. Identification and SAR exploration of a novel series of Legumain inhibitors. Bioorg Med Chem Lett. 2019 Jun 15;29 (12) :1546-1548.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
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