DA 4626
DA 4626 is a competitive H2-histamine receptor antagonist. DA 4626 inhibits adenylate cyclase activity with a KB value of 40 nM[1].
Product Specifications
CAS Number
83184-14-9
UNSPSC
12352005
Target
Adenylate Cyclase; Histamine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/da-4626.html
Smiles
CC(/N=C/NC1=CC=C(C2=CN=CN2)C=C1)(C)C
Molecular Formula
C14H18N4
Molecular Weight
242.32
References & Citations
[1]Micheletti R, et al. Evaluation of novel compounds interacting with H2-histamine receptors: effect on histamine-sensitive adenylate cyclase activity in guinea-pig gastric mucosa. Agents Actions. 1985 Jul;16 (5) :291-4.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
H2 Receptor
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