GCPII-IN-1
GCPII-IN-1 (Compound 2) is a GCPII (also known as PSMA) inhibitor scaffold with a Ki of 44.3 nM. GCPII-IN-1 can be used in the research of prostate cancer[1].
Product Specifications
CAS Number
[1025796-32-0]
UNSPSC
12352211
Target
Carboxypeptidase; PSMA
Type
Reference compound
Related Pathways
Immunology/Inflammation; Metabolic Enzyme/Protease
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/gcpii-in-1.html
Purity
99.83
Solubility
DMSO : 50 mg/mL (ultrasonic)
Smiles
NCCCC[C@@H](C(O)=O)NC(N[C@H](C(O)=O)CCC(O)=O)=O
Molecular Formula
C12H21N3O7
Molecular Weight
319.31
References & Citations
[1]Jan Tykvart, et al. Rational design of urea-based glutamate carboxypeptidase II (GCPII) inhibitors as versatile tools for specific drug targeting and delivery. Bioorg Med Chem. 2014 Aug 1;22 (15) :4099-108.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Curated Selection
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