GPR88 agonist 2
GPR88 agonist 2 (compound 53) is a potent and brain-penetrantGPR88 agonist with an EC50 value of 14 µM in GPR88 cAMP functional assay[1].
Product Specifications
CAS Number
2821859-71-4
UNSPSC
12352005
Target
GPR88
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease; Others
Assay Protocol
https://www.medchemexpress.com/gpr88-agonist-2.html
Purity
99.57
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
CNC(C(N=N1)=CN1C[C@@H](C2=CC=C(C=C2)OC[C@@H](C)CC)NC([C@H](C3=CC=CC=C3)C)=O)=O
Molecular Formula
C26H33N5O3
Molecular Weight
463.57
References & Citations
[1]Rahman MT, et al. Evaluation of Amide Bioisosteres Leading to 1,2,3-Triazole Containing Compounds as GPR88 Agonists: Design, Synthesis, and Structure-Activity Relationship Studies. J Med Chem. 2021 Aug 26;64 (16) :12397-12413.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
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