What is the catalog number for UFP-101?

The catalog number for UFP-101 is HY-P1299.

What sizes are available for UFP-101?

UFP-101 is available in the following size(s): 1 Each.

UFP-101 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures UFP-101?

UFP-101 is manufactured by QuantiMol.

What is the estimated delivery time for UFP-101?

Estimated delivery time for UFP-101 is approximately 15 business day(s), depending on your location.

Where can I find the safety data sheet (SDS/MSDS) for UFP-101?

The safety data sheet for UFP-101 is available here: http://file.medchemexpress.com/batch_PDF/HY-P1299/.

UFP-101

UFP-101 is a potent, selective, and competitive antagonist of the NOP receptor, with a pKi of 10.24. UFP-101 displays >3000-fold selectivity over δ, μ and κ opioid receptors. UFP-101 shows antidepressant-like effect[1][2].

Product Specifications

CAS Number

849024-68-6

UNSPSC

12352209

Target

Opioid Receptor

Type

Peptides

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/ufp-101.html

Solubility

10 mM in DMSO

Smiles

[C@H](CC1=CC=CC=C1)(C(N[C@H](C(NCC(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@@H](CCC(N)=O)C(N)=O)=O)CC(N)=O)=O)CCCCN)=O)CCCNC(=N)N)=O)CCCCN)=O)CCCNC(=N)N)=O)C)=O)CO)=O)CCCCN)=O)CCCNC(=N)N)=O)C)=O)=O)[C@@H](C)O)=O)NC(CNC(CNC(CNCC2=CC=CC=C2)=O)=O)=O

Molecular Formula

C82H138N32O21

Molecular Weight

1908.17

References & Citations

[1]Calo G, et al. [Nphe1, Arg14, Lys15]nociceptin-NH2, a novel potent and selective antagonist of the nociceptin/orphanin FQ receptor. Br J Pharmacol. 2002;136 (2) :303-311.|[2]Gavioli EC, et al. Blockade of nociceptin/orphanin FQ-NOP receptor signalling produces antidepressant-like effects: pharmacological and genetic evidences from the mouse forced swimming test. Eur J Neurosci. 2003;17 (9) :1987-1990.