Protease-Activated Receptor-4

Protease-Activated Receptor-4 is the agonist of proteinase-activated receptor-4 (PAR4) .

Product Specifications

CAS Number

[245443-52-1]

UNSPSC

12352209

Target

Protease Activated Receptor (PAR)

Type

Peptides

Related Pathways

GPCR/G Protein

Field of Research

Others

Assay Protocol

https://www.medchemexpress.com/Protease-Activated_Receptor-4.html

Purity

95.03

Solubility

10 mM in DMSO|H2O : 50 mg/mL (ultrasonic)

Smiles

O=C(N)[C@H](CC1=CC=CC=C1)NC([C@H](CCCCN)NC(CNC([C@H]2N(C([C@H](CC3=CC=C(C=C3)O)NC(CN)=O)=O)CCC2)=O)=O)=O

Molecular Formula

C33H46N8O7

Molecular Weight

666.77

References & Citations

[1]Moschonas IC, et al. Molecular requirements involving the human platelet protease-activated receptor-4 mechanism of activation by peptide analogues of its tethered-ligand. Platelets. 2017 Mar 7:1-10. doi: 10.1080/09537104.2017.1282607. [Epub ahead of print]|[2]Huang SC, et al. Proteinase-activated receptor-1 (PAR1) and PAR2 mediate relaxation of guinea pig internal anal sphincter. Regul Pept. 2014 Feb 10;189:46-50.