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MRGPRX4 modulator-1

Product Specifications

UNSPSC Description

MRGPRX4 modulator-1 (compound 31-2) is a potent mas-related g-protein receptor X4 (MRGPR X4) modulator, with antagonist activity of IC50 [1].

Target Antigen

Mas-related G-protein-coupled Receptor (MRGPR)

Type

Reference compound

Related Pathways

GPCR/G Protein

Applications

COVID-19-immunoregulation

Field of Research

Inflammation/Immunology

Assay Protocol

https://www.medchemexpress.com/mrgprx4-modulator-1.html

Solubility

DMSO : 100 mg/mL (ultrasonic)

Smiles

O=C(C1=NC(COC2=CC=C(C(F)(F)F)C=C2Cl)=CC(CC)=C1)O

Molecular Weight

359.73

References & Citations

[1]Adam YEAGER, et al. Modulators of mas-related g-protein receptor x4 and related products and methods. WO2020198537 (compound 31-2).

Shipping Conditions

Room Temperature

Product Datasheet

http://file.medchemexpress.com/batch_PDF/HY-145997/MRGPRX4-modulator-1-DataSheet-MedChemExpress.pdf

Product MSDS

http://file.medchemexpress.com/batch_PDF/HY-145997/MRGPRX4-modulator-1-SDS-MedChemExpress.pdf

Clinical Information

No Development Reported

CAS Number

2492596-61-7

Available Sizes

Curated Selection

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