MDA77
MDA77 is a CB2 inverse agonist with an EC50 of 5.82 nM, showing selectivity for human CB2 and no activity on CB1[1].
Product Specifications
CAS Number
1103774-21-5
UNSPSC
12352005
Target
Cannabinoid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Inflammation/Immunology; Neurological Disease
Assay Protocol
https://www.medchemexpress.com/mda77.html
Smiles
O=C(N/N=C1C(N(CCCCC)C2=C\1C=CC(OC)=C2)=O)C3=CC=CC=C3
Molecular Formula
C21H23N3O3
Molecular Weight
365.43
References & Citations
[1]Philippe Diaz, et al. 6-Methoxy-N-alkyl isatin acylhydrazone derivatives as a novel series of potent selective cannabinoid receptor 2 inverse agonists: design, synthesis, and binding mode prediction. J Med Chem. 2009 Jan 22;52 (2) :433-44.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
K2685402 1.0 µg DNA
ZNF79 sgRNA CRISPR Lentivector (Human) (Target 1)
Sign In for Pricing
View Details 