MDA77

MDA77 is a CB2 inverse agonist with an EC50 of 5.82 nM, showing selectivity for human CB2 and no activity on CB1[1].

Product Specifications

CAS Number

[1103774-21-5]

UNSPSC

12352005

Target

Cannabinoid Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Inflammation/Immunology; Neurological Disease

Assay Protocol

https://www.medchemexpress.com/mda77.html

Smiles

O=C(N/N=C1C(N(CCCCC)C2=C\1C=CC(OC)=C2)=O)C3=CC=CC=C3

Molecular Formula

C21H23N3O3

Molecular Weight

365.43

References & Citations

[1]Philippe Diaz, et al. 6-Methoxy-N-alkyl isatin acylhydrazone derivatives as a novel series of potent selective cannabinoid receptor 2 inverse agonists: design, synthesis, and binding mode prediction. J Med Chem. 2009 Jan 22;52 (2) :433-44.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Available Sizes

Curated Selection

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